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Carteolol









Carteolol


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Carteolol
Carteolol skeletal.svg
Clinical data
Trade names Ocupress

AHFS/Drugs.com
 Micromedex Detailed Consumer Information
MedlinePlus a601078
Pregnancy
category


  • US: C (Risk not ruled out)


Routes of
administration		 Eye drops
ATC code

  • C07AA15 (WHO) S01ED05 (WHO)
Legal status
Legal status

  • In general: ℞ (Prescription only)

Pharmacokinetic data
Bioavailability 85%
Metabolism
Hepatic, active with 8-hydrocarteolol
Elimination half-life
 6–8 hours
Excretion
Renal (50-70%)
Identifiers
CAS Number
  • 51781-06-7

PubChem CID
  • 2583
IUPHAR/BPS
  • 7142
DrugBank

  • DB00521 ☑Y
ChemSpider

  • 2485 ☑Y
UNII
  • 8NF31401XG
KEGG

  • D07624 ☑Y
ChEBI

  • CHEBI:3437 ☑Y
ChEMBL

  • ChEMBL839 ☑Y
Chemical and physical data
Formula
C16H24N2O3
Molar mass 292.373 g/mol
3D model (JSmol)
  • Interactive image
Chirality Racemic mixture

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Carteolol[a] is a non-selective beta blocker used to treat glaucoma.


It has been found to act as a serotonin 5-HT1A and 5-HT1B receptor antagonist in addition to being a beta blocker.[1]



Notes[edit]





  1. ^ Trade names include Cartrol, Ocupress, Teoptic, Arteolol, Arteoptic, Calte, Cartéabak, Carteol, Cartéol, Cartrol, Elebloc, Endak, Glauteolol, Mikelan, Poenglaucol, and Singlauc.




References[edit]





  1. ^ Langlois M, Brémont B, Rousselle D, Gaudy F (1993). "Structural analysis by the comparative molecular field analysis method of the affinity of beta-adrenoreceptor blocking agents for 5-HT1A and 5-HT1B receptors". Eur. J. Pharmacol. 244 (1): 77–87. doi:10.1016/0922-4106(93)90061-d. PMID 8093601..mw-parser-output cite.citation{font-style:inherit}.mw-parser-output q{quotes:"""""""'""'"}.mw-parser-output code.cs1-code{color:inherit;background:inherit;border:inherit;padding:inherit}.mw-parser-output .cs1-lock-free a{background:url("//upload.wikimedia.org/wikipedia/commons/thumb/6/65/Lock-green.svg/9px-Lock-green.svg.png")no-repeat;background-position:right .1em center}.mw-parser-output .cs1-lock-limited a,.mw-parser-output .cs1-lock-registration a{background:url("//upload.wikimedia.org/wikipedia/commons/thumb/d/d6/Lock-gray-alt-2.svg/9px-Lock-gray-alt-2.svg.png")no-repeat;background-position:right .1em center}.mw-parser-output .cs1-lock-subscription a{background:url("//upload.wikimedia.org/wikipedia/commons/thumb/a/aa/Lock-red-alt-2.svg/9px-Lock-red-alt-2.svg.png")no-repeat;background-position:right .1em center}.mw-parser-output .cs1-subscription,.mw-parser-output .cs1-registration{color:#555}.mw-parser-output .cs1-subscription span,.mw-parser-output .cs1-registration span{border-bottom:1px dotted;cursor:help}.mw-parser-output .cs1-hidden-error{display:none;font-size:100%}.mw-parser-output .cs1-visible-error{font-size:100%}.mw-parser-output .cs1-subscription,.mw-parser-output .cs1-registration,.mw-parser-output .cs1-format{font-size:95%}.mw-parser-output .cs1-kern-left,.mw-parser-output .cs1-kern-wl-left{padding-left:0.2em}.mw-parser-output .cs1-kern-right,.mw-parser-output .cs1-kern-wl-right{padding-right:0.2em}




External links[edit]




  • El-Kamel A, Al-Dosari H, Al-Jenoobi F (2006). "Environmentally responsive ophthalmic gel formulation of carteolol hydrochloride". Drug Deliv. 13 (1): 55–9. doi:10.1080/10717540500309073. PMID 16401594.


  • Kuwahara K, Oizumi N, Fujisawa S, Tanito M, Ohira A (2005). "Carteolol hydrochloride protects human corneal epithelial cells from UVB-induced damage in vitro". Cornea. 24 (2): 213–20. doi:10.1097/01.ico.0000141232.41343.9d. PMID 15725891.


  • Trinquand C, Romanet J, Nordmann J, Allaire C (2003). "[Efficacy and safety of long-acting carteolol 1% once daily. A double-masked, randomized study]". J Fr Ophtalmol. 26 (2): 131–6. PMID 12660585.

















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